Key Pharmacologic Principles and Drug-Drug Interactions in HIV Patient Care
Summary
- Absorption, Distribution, Metabolism, and Elimination
- Antiretrovirals undergo pharmacokinetic transformation during absorption, distribution, metabolism, and elimination
- Most clinically relevant drug interactions involving antiretrovirals occur because of alterations in drug-metabolizing enzyme activity
- Renal elimination is not a common cause of antiretroviral drug interactions
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Keywords: Drug-Drug Interactions, Pharmacokinetics